奥巴克拉是一种 BCL-2 家族拮抗剂,结合 BCL-2,Ki 约为 220 nM.Obatoclax 抑制所有 BCL-XL,MCL-1,BCL-w,A1 和 BCL-b 的相互作用 (Ki≈1-7 μM).
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95+% CAS No.:69778-83-2
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