艾代拉里斯是一种有效的选择性的 p110δ 抑制剂,IC50 为 2.5 nM,比作用于其他I类 PI3K 酶 (抑制 p110α,p110β 和 p110γ,IC50 分别为 820,565 和 89 nM) 选择性高 40 到 300 倍.它是一种用于治疗某些血液系统恶性肿瘤的药物.该物质起磷酸肌醇3激酶抑制剂的作用;更具体地说,它阻断P110δ,即磷酸肌醇3激酶的δ同工酶.
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≥98.0% CAS No.:87-42-3
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97% CAS No.:870281-83-7
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