达拉非尼是ATP竞争型的 Raf 抑制剂,抑制 C-Raf 和 B-RafV600E 的 IC50 分别为 5 nM 和 0.6 nM,是一种用于治疗与突变基因BRAF相关的癌症的药物,作为相关酶B-RAF的抑制剂,在细胞生长的调节中起着一定的作用.
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