多巴胺受体是一类G蛋白偶联受体,在脊椎动物中枢神经系统(CNS)中是突出的.神经递质多巴胺是多巴胺受体的主要内源性配体.多巴胺受体参与许多神经过程,包括动机、快感、认知、记忆、学习和精细运动控制,以及神经内分泌信号的调节.多巴胺受体信号转导异常和多巴胺能神经功能异常与多种神经精神疾病有关.因此,多巴胺受体是常见的神经药物靶点,抗精神病药物通常是多巴胺受体拮抗剂,而精神刺激剂通常是多巴胺受体
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