贝曲西班是一种口服有效的选择性直接因子(fXa)抑制剂,IC50 为 1.5 nM,是一种口服抗凝药,其作用是直接因子Xa抑制剂,是用于预防因急性内科疾病住院的成年人静脉血栓形成的药物,该疾病由于活动受限和易发生血栓栓塞并发症.
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