奥扎莫德是一种有效的选择性 S1P1 和 S1P5 受体激动剂,在[35S]-GTPγS 结合实验中,EC50 分别为 410±160 pM 和 11±4.3 nM,是一种研究性免疫调节药物,目前正处于治疗复发性多发性硬化症(RMS)和溃疡性结肠炎(UC)的III期临床试验.它作为一个鞘氨醇-1-磷酸(S1P)受体激动剂,隔离淋巴细胞到外周淋巴器官和远离其慢性炎症部位.
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98% CAS No.:15115-60-3
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≥98% CAS No.:196929-78-9
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98% CAS No.:258273-31-3
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97+% CAS No.:60899-34-5
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