雷多替尼是酪氨酸激酶Bcr-Abl1新型选择性抑制剂,对野生型Bcr-Abl1的IC50值为34nM,是一种治疗不同类型癌症的药物,最显著的是费城染色体阳性(Ph+)慢性髓细胞白血病(CML),对其他Bcr-Abl酪氨酸激酶抑制剂(如pa)耐药或不耐受.对伊马替尼耐药或耐受.
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