帕利替尼是一种有效的野生型 JAK2 和 JAK2V617F 突变型抑制剂,IC50 分别为 23 nM 和 19 nM.Pacritinib 也抑制 FLT3及其突变型FLT3D835Y,IC50 分别为 22 nM 和 6 nM.它是一种正在开发用于治疗骨髓纤维化的大环JANUS激酶抑制剂.它主要抑制JANK激酶2(JAK2)和FMS样酪氨酸激酶3(FLT3).
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≥98% CAS No.:97-51-8
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SKU-Pack Size Availability Price(¥) Quantity R002359-5g In-Stock(Shanghai or CA Irwindale) R002359-5g In-Stock(Shanghai or CA Irwindale) R002359-100g In-Stock(Shanghai or CA Irwindale) R002359-25g In-Stock(Shanghai or CA Irwindale) R002359-500g In-Stock(Shanghai or CA Irwindale) R002359-5g In-Stock(Shanghai or CA Irwindale) R002359-100g In-Stock(Shanghai or CA Irwindale) R002359-25g In-Stock(Shanghai or CA Irwindale) R002359-500g In-Stock(Shanghai or CA Irwindale) R002359-10g In-Stock(Shanghai or CA Irwindale) R002359-25g In-Stock(Shanghai or CA Irwindale) R002359-100g In-Stock(Shanghai or CA Irwindale) R002359-500g In-Stock(Shanghai or CA Irwindale) R002359-1000g In-Stock(Shanghai or CA Irwindale) -
≥98% CAS No.:87199-15-3
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SKU-Pack Size Availability Price(¥) Quantity R421031-5g In-Stock(Shanghai or CA Irwindale) R421031-1g In-Stock(Shanghai or CA Irwindale) R421031-1g In-Stock(Shanghai or CA Irwindale) R421031-25g In-Stock(Shanghai or CA Irwindale) R421031-5g In-Stock(Shanghai or CA Irwindale) R421031-100g In-Stock(Shanghai or CA Irwindale) R421031-1g In-Stock(Shanghai or CA Irwindale) R421031-25g In-Stock(Shanghai or CA Irwindale) R421031-5g In-Stock(Shanghai or CA Irwindale) R421031-100g In-Stock(Shanghai or CA Irwindale) R421031-10g In-Stock(Shanghai or CA Irwindale) R421031-25g In-Stock(Shanghai or CA Irwindale) R421031-100g In-Stock(Shanghai or CA Irwindale) R421031-500g In-Stock(Shanghai or CA Irwindale)