奥普唑米是口服活性第二代蛋白酶体抑制剂,能抑制20S proteasome(20S蛋白酶体)β5/LMP7的CT-L活性,IC50为36 nM/82 nM,它有选择性地抑制组成蛋白酶体(PSMb5)和免疫蛋白酶体(LMP7)的糜蛋白酶样活性.
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97% CAS No.:51293-47-1
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98% CAS No.:40004-69-1
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