乐伐替尼是一种口服,多靶点酪氨酸激酶抑制剂,抑制 VEGFR2(KDR) 和 VEGFR3(Flt-4) 的 IC50 分别为 4 和 5.2 nM,是一种抗癌药物,用于治疗某些类型的甲状腺癌,也可用于治疗其他癌症.
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