戈勒特隆是一种多功能的抗雄激素,是 CYP17 抑制剂,在去势抵抗性前列腺癌中,IC50 为 47 nM,是一种甾体抗雄激素,是用于治疗前列腺癌的药物.它具有独特的双重作用机制,既是雄激素受体拮抗剂,又是CYP17A1抑制剂,后者阻止雄激素的生物合成.
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≥98% CAS No.:51-17-2
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