氟洛克生是一种有效的α2-肾上腺素能受体拮抗剂(pKB=7.9),具有优良的α2/α1选择性(2630倍),是结构家族中唯一研究得比较多的不拮抗咪唑啉受体变异体的a2拮抗剂.该化合物口服后具有中枢α2-肾上腺素能受体拮抗剂活性,在20世纪80年代初被葛兰素公司专利为抗抑郁药.
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95% CAS No.:1660-93-1
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97% CAS No.:90365-74-5
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