司马西特是一种 γ-secretase 抑制剂,抑制 β-amyloid (Aβ42),Aβ38 和 Aβ40,IC50 分别为 10.9,12 和 12.1 nM.也抑制 Notch,IC50 为 14.1 nM,是一种用于阿尔茨海默病的因果疗法的候选药物.
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97% CAS No.:17407-55-5
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